Palladium-catalyzed ortho-acylation of 2-benzyl-1,2,3-triazoles with aldehydes.
نویسندگان
چکیده
A palladium-catalyzed ortho-acylation of 2-benzyl-1,2,3-triazoles with aldehydes as an acyl source was developed. A wide variety of ketones containing 1,2,3-triazoles were obtained in good to excellent yields. This methodology provides a convenient access to the acylation of 2-substituted-1,2,3-triazoles.
منابع مشابه
Palladium-catalyzed ortho-C-H alkenylation of 2-benzyl-1,2,3-triazoles.
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 12 38 شماره
صفحات -
تاریخ انتشار 2014